Energy bar Number:7,037,531 from the United States Patent and Trademark Office (PTO) owispatent An energy multi-saccharide food product including: a saccharide component including 5 to 20% w/w galactose; to 25% w/w creatine; and optional further ingredients selected from: carbohydrate, fibre and fat.<H Energy, bar, Energy, bar, 7037531.html, Patent, pto, 7037531

Title: Energy bar

Abstract: An energy multi-saccharide food product including: a saccharide component including 5 to 20% w/w galactose; to 25% w/w creatine; and optional further ingredients selected from: carbohydrate, fibre and fat.

Patent Number: 7,037,531 Issued on 05/02/2006 to King, et al.

Inventors: King; Roderick Frederick Gerardus Joseph (West Yorkshire, GB); Gale; Richard William (North Yorkshire, GB); Lester; Simon Edmund George (London, GB)
Assignee: Galactogen Products Limited (London, GB)

Appl. No.: 379160

Filed: March 3, 2003

Related U.S. Patent Documents


Application Number	Filing Date	Patent Number	Issue Date
09692516	Oct., 2000	6585999

Current U.S. Class: 424/725 ; 536/1.11

Current International Class: A61K 35/78 (20060101); C07H 1/00 (20060101)

Field of Search: 424/479 524/58 426/615,658,660

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3753725	August 1973	Williams et al.
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5401524	March 1995	Burkes et al.
5487894	January 1996	Kovacs
5587190	December 1996	Guezennec et al.
5612074	March 1997	Leach
5726146	March 1998	Almada et al.
5780094	July 1998	King
5843921	December 1998	Kaufman
6787177	September 2004	Crandall et al.
2003/0082287	May 2003	Wolt et al.

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Primary Examiner: Leith; Patricia
Attorney, Agent or Firm: Beyer Weaver & Thomas LLP

Parent Case Text

"This is a Continuation application of prior application Ser. No. 09/692,516, filed Oct. 18, 2000 now U.S. Pat. No. 6,585,999, which claims priority of United Kingdom Application No.: 9924650.6, filed Oct. 19, 1999, filed on which designated the United States, the disclosures of which are incorporated herein by reference."

Claims

What is claimed is:

1. An energy multi-saccharide food product, comprising: no more than 15% by total weight dried fruit; a saccharide component comprising 3 to 37% by total weight free galactose monosaccharide; and 5 to 10% by total weight fiber.

2. The food product of claim 1, further comprising up to 25% by total weight creatine.

3. The food product of claim 2, wherein the amount of creatine is 10 to 25%.

4. The food product of claim 3, wherein the creatine is encapsulated as granules or powder.

5. The food product of claim 4, wherein the creatine is microencapsulated.

6. The food product of claim 3, wherein the creatine is contained in a layer separate from other ingredients of the food product.

7. The food product of claim 1, wherein the amount of galactose is 5 to 20%.

8. The food product of claim 1, wherein the saccharide component comprises glucose.

9. The food product of claim 8, wherein the saccharide component comprises equal amounts of galactose and glucose.

10. The food product of claim 8, wherein the amount of galactose is greater than the amount of glucose.

11. The food product of claim 1, having an outermost layer of hard sugar comprising galactose or a mixture of galactose and sucrose.

12. A food product as claimed in claim 1, wherein the saccharide component comprises fructose.

13. A food product as claimed in claim 1, wherein the saccbaride component comprises maltodextrin.

14. A food product as claimed in claim 1, wherein the saccharide component comprises maltodextrin and fructose.

15. A method for replenishing glycogen reserves in a subject, the method comprising: administering to the subject the food product of claim 1.

16. The method of claim 15, wherein the replenished glycogen reserves are in liver.

17. The method of claim 15, wherein the replenished glycogen reserves are in muscle.

18. The method of claim 15, wherein the food product is orally administered.

Description

This invention relates to high energy multi-saccharide food products containing the substance galactose, which find use as an ergogenic aid, particularly but not exclusively for persons participating in sports or other forms of exercise. The products of this invention also find use in cases of hunger or fatigue in the general population.

Exercise makes excessive demands on substrates both within and external to the muscle. Carbohydrates are especially important as precursors of glycogen both in liver and muscle and as an energy source which can be used immediately. Accordingly there is a need for a short term energy supply during anaerobic and aerobic conditions. It is also a requirement for carbohydrates which serve as precursors either directly or indirectly for synthesis of glycogen in liver and muscle. Muscle cannot function efficiently or at a high level of power output if reserves of glycogen are low or sub-optimal. Depletion of glycogen in athletes results in poor performance and poor efficiency. Use of specific carbohydrates as an ergogenic aid has been proved to increase or maintain the stores of glycogen and availability of blood glucose.

The food products of this invention may comprise chewable or edible bars, sweets, cookies, biscuits, lozenges or chewing gum. Chewable or edible bars are preferred.

According to the present invention a high energy multi-saccharide food product comprises a saccharide component including 3 to 37% w/w galactose, 0 to 25% w/w of creatine and optional further ingredients selected from carbohydrate; fibre and fat.

Amounts and percentages in this specification are by weight unless indicated otherwise and are selected to total 100%.

The amount of galactose is preferably 5 to 20%, more preferably 5 to 15%.

The saccharide component also includes glucose. In a first preferred embodiment equal amounts of glucose and galactose are provided. In a second preferred embodiment the amount of galactose is greater than the amount of glucose.

Use of galactose affords several advantages. It is not insulogenic, that is it does not itself induce an insulin response, hence its use is associated with less of an insulin response than the equivalent mass of glucose. Products in accordance with this invention may be used by diabetics or persons who ae intolerant to lactose. Galactose can be used rapidly by the liver for synthesis of glycogen or glucose. It is less likely to cause dental erosion than other sugars.

Use of creatine is optional. Preferred embodiments of the invention incorporate 10 to 25% creatine. The use of creatine is preferably such that the conversion to creatinine is inhibited. This conversion is a natural equilibrium. Creatinine is rapidly excreted by-the kidneys. In order to minimise or prevent conversion to creatinine it is preferred that the creatine is encapsulated as granules or powder in a dry water-impervious shell. Micro-encapsulation is preferred. In this way the creatine is released in the stomach by dissolution. Alternatively the creatine may be isolated from the moist part of an edible bar by formulation in layers alternatively or in addition to encapsulation. For example the creatine may be contained in a separate layer of the food bar or lozenge.

Food products in accordance with this invention are useful in general cases of creatine depletion, for example in vegetarians or individuals where build-up of muscle function is needed or is clinically advisable.

Exercise makes excessive demands on substrates both within and external to muscle. Creatine phosphate is derived from both dietary creatine and from endogenous synthesis. Creatine phosphate is essential for short term energy supply during anaerobic conditions and also for energy transfer from mitochondria to contractile muscle. Muscle cannot function efficiently or at a high level of power output if reserves of creatine are low or sub-optimal. Depletion of creatine in athletes causes poor performance and poor efficiency.

Galactose may be provided as a pure ingredient which is mixed with glucose, starch and other ingredients during manufacture. Alternatively a glucose-galactose syrup such as may be prepared by hydrolysis of lactose may be employed. The amount of galactose in such a syrup may be supplemented by additional pure galactose.

Use of fibre in the bar is advantageous because different fibre products influence the release of sugars, affect the binding of various components and advantageously delay digestion. An amount of 0 to 5% may be employed. Furthermore the galactose or galactose-glucose syrup may be absorbed onto the fibre prior to manufacture. In this way the absorption of galactose may be retarded.

In an alternative embodiment the food products may have an external coating containing galactose in order to facilitate rapid absorption of galactose.

Formulations having a higher concentration of galactose are preferred in order to enhance galactose up-take by the liver and rapid production of glycogen. Increased amounts of galactose decrease the amount of lipid manufactured from glucose. Galactose is not a direct fat precursor. This is advantageous as lipids do not afford a rapid energy source.

The invention is further described by means of example but not in any limitative sense.

The following Tables and Examples list the ingredients of compositions of food products in accordance with this invention. These products may be manufactured into bars, sweets or lozenges using conventional methods.

In a layered arrangement the creatine powder or aggregate may be covered with a hard dry sugar layer. Alternatively or in addition a chocolate containing layer may be used as a moisture barrier. The creatine containing layer may be provided as a larninar cylindrical layer disposed within the bar as the inner layer. In this way the creatine containing component may be encapsulated. Alternatively or in addition ingredients such as fibre, nuts and dried fruit may be layered onto the creatine to form a laminate. The fibre layer may incorporate syrup to form a composite layer.

The outermost layer of the bar or other food product may comprise a single thin layer of hard sugar for example composed of galactose or a mixture of galactose with glucose or sucrose. Such an arrangement of the sugar layer dissolves rapidly when portions of the bar pass into the stomach.

In alternative food products the creatine powder or aggregate may be covered with a hard sugar mixture, chocolate or both to form particles with a mass of 100 to 500 mg. These can be combined with the remaining ingredients to form dispersed units within the matrix, for example as chocolate chips within a cookie. Such an encapsulated arrangement may incorporate layers as previously described.

The following tables contain general ranges of preferred ingredients.

TABLE-US-00001 TABLE 1 Ingredient Range (% w/w) Comments Carbohydrate 50 75 Mono, di, oligosaccharides, syrup etc. Fat 0 10 Saturated and unsaturated Fibre 0 10 Creatine 0 25 As monohydrate Protein 0 15 Vitamins 50 100% of RDA Full range Galactose 5 20 Dried Fruit 0 15 Seeds and Nuts 0 15 Glucose 0 10 Flavours As necessary Stabilisers 1 3 Water 0 30

TABLE-US-00002 TABLE 2 Example 1 Example 2 Example 3 Example 4 Example 5 Example 6 Cornstarch 20 g 10 g 20 g 10 g 10 g 8 g Maltodextrin 20 g 10 g 20 g 10 g 10 g 8 g Raw cane sugar 2 g 2 g 2 g 2 g 2 g 2 g Fructose 3 g 3 g 3 g 3 g 3 g -- Refined cane sugar 5 g 5 g 5 g 5 g 5 g -- Glucose 5 g 5 g -- -- 5 g 5 g Galactose 5 g 5 g -- -- 5 g 5 g Glucose/Galactose -- -- 10 g 10 g -- -- syrup Fat 10 g 10 g 10 g 10 g 10 g 5 g Fibre 5 g 5 g 5 g 5 g 5 g 5 g Creatine -- 20 g -- 20 g -- 20 g Vitamins 1 g 1 g 1 g 1 g 1 g 1 g Protein 10 g 10 g 10 g 10 g 10 g 7 g Flavours 1 g 1 g 1 g 1 g 1 g 1 g Stabilisers 2 g 2 g 2 g 2 g 2 g 2 g Water 11 g 11 g 11 g 11 g 11 g 11 g Fruit -- -- -- -- 10 g 10 g Seeds and Nuts -- -- -- -- 10 g 10 g Example 7 Example 8 Example 9 Example 10 Example 11 Example 12 Cornstarch 20 g 10 g 20 g 10 g 10 g 8 g Maltodextrin 20 g 10 g 20 g 10 g 10 g 8 g Raw cane sugar 2 g 2 g 2 g 2 g 2 g 2 g Fructose 3 g 3 g 3 g 3 g 3 g -- Refined cane 5 g 5 g 5 g 5 g 5 g -- sugar Glucose 5 g 5 g -- -- 5 g 5 g Galactose 5 g 5 g -- -- 5 g 5 g Glucose/Galactose -- -- 10 g 10 g -- -- syrup Fat 10 g 10 g 10 g 10 g 10 g 5 g Fibre 5 g 5 g 5 g 5 g 5 g 5 g Creatine -- 20 g -- 20 g -- 20 g Vitamins 1 g 1 g 1 g 1 g 1 g 1 g Protein 10 g 10 g 10 g 10 g 10 g 7 g Flavours 1 g 1 g 1 g 1 g 1 g 1 g Stabilisers 2 g 2 g 2 g 2 g 2 g 2 g Water 5 g 5 g 5 g 5 g 5 g 5 g Fruit 3 g 3 g 3 g 3 g 13 g 13 g Seeds and Nuts 3 g 3 g 3 g 3 g 13 g 13 g Example 13 Example 14 Example 15 Example 16 Example 17 Example 18 Cornstarch 15 g 5 g 15 g 5 g 5 g 8 g Maltodextrin 15 g 5 g 15 g 5 g 5 g 8 g Raw cane sugar 2 g 2 g 2 g 2 g 2 g 2 g Fructose 3 g 3 g 3 g 3 g 3 g -- Refined cane 5 g 5 g 5 g 5 g 5 g -- sugar Glucose 5 g 5 g -- -- 5 g 5 g Galactose 5 g 5 g -- -- 5 g 5 g Glucose/Galactose -- -- 10 g 10 g -- -- syrup Fat 10 g 10 g 10 g 10 g 18 g 3 g Fibre 5 g 5 g 5 g 5 g 2 g 2 g Creatine -- 20 g -- 20 g -- 20 g Vitamins 1 g 1 g 1 g 1 g 1 g 1 g Protein 5 g 5 g 5 g 5 g 5 g 2 g Flavours 1 g 1 g 1 g 1 g 1 g 1 g Stabilisers 2 g 2 g 2 g 2 g 2 g 2 g Water 20 g 20 g 20 g 20 g 20 g 20 g Fruit 3 g 3 g 3 g 3 g 13 g 13 g Seeds and Nuts 3 g 3 g 3 g 3 g 8 g 8 g

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